Table 9. Reference Summary: σR Binding (679, 680).
| Drug | Target tissue |
|---|---|
| (+)-pentazocine [PTZ] | Sigma1 Sigma2 ligands |
| Haloperidol [Haldol®] | Sigma1 Sigma2 ligands |
| 1,3 di-o-tolyl-guanidine [DTG] | Sigma1 Sigma2 ligands |
| (+)-3-PPP [preclamol] | Sigma1 Sigma2 ligands |
| (+)-SKF 10,047 | Sigma1 Sigma2 ligands |
| (+)-pentazocine [PTZ] | Sigma1 Sigma2 ligands |
| Phencyclidine | Sigma1 Sigma2 ligands |
| Dextromethorphan [DEX] | Sigma1 ligands |
| (+)-cyclazocine | Sigma1 ligands |
| BD1047 | Sigma2 ligands |
| BD1063 | Sigma2 ligands |