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. 2015 Jun 9;36(4):327–388. doi: 10.3109/10799893.2015.1015737

Table 9. Reference Summary: σR Binding (679, 680).

Drug Target tissue
(+)-pentazocine [PTZ] Sigma1 Sigma2 ligands
Haloperidol [Haldol®] Sigma1 Sigma2 ligands
1,3 di-o-tolyl-guanidine [DTG] Sigma1 Sigma2 ligands
(+)-3-PPP [preclamol] Sigma1 Sigma2 ligands
(+)-SKF 10,047 Sigma1 Sigma2 ligands
(+)-pentazocine [PTZ] Sigma1 Sigma2 ligands
Phencyclidine Sigma1 Sigma2 ligands
Dextromethorphan [DEX] Sigma1 ligands
(+)-cyclazocine Sigma1 ligands
BD1047 Sigma2 ligands
BD1063 Sigma2 ligands