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. 2016 Jun 20;11(6):e0157039. doi: 10.1371/journal.pone.0157039

Table 1. Lopinavir (200 mg)/Ritonavir (50 mg) drug sources and characteristics.

Site Lot No. Manufacturer Country Trade name WHO Prequal. Expiry date Identification % of label amount Uniformity of mass, % Dissolution, % (LPV/RTV)
Min Max Min Max
001 W570041 GPO THA Lopinavir/Ritonavir NO 21 Jan 16 Positive 102.1/100.8 -1.20 1.64 97.6/98.8 98.2/99.7
002 W560404 GPO THA Lopinavir/Ritonavir NO 13 Jul 15 Positive 103.2/102.4 -1.28 1.48 98.1/100.8 99.1/102.2
003 W570169 GPO THA Lopinavir/Ritonavir NO 17 Mar 16 Positive 102.1/103.6 -1.11 1.25 99.1/100.0 101.2/103.1
004 W570175 GPO THA Lopinavir/Ritonavir NO 17 Mar 16 Positive 101.0/103.3 -2.22 2.08 97.7/99.0 101.9/102.5
005 W570450 GPO THA Lopinavir/Ritonavir NO 17 Jul 16 Positive 99.4/101.8 -2.16 1.07 97.5/99.0 101.3/102.8
006 W560432 GPO THA Lopinavir/Ritonavir NO 23 Jul 15 Positive 99.0/103.0 -2.10 1.87 98.5/100.3 102.6/104.6
007 W570457 GPO THA Lopinavir/Ritonavir NO 20 Jul 16 Positive 98.6/101.5 -1.74 2.05 98.7/95.0 99.8/97.0
008 W570152 GPO THA Lopinavir/Ritonavir NO 10 Mar 16 Positive 99.4/101.4 -2.09 1.76 96.2/99.0 98.7/102.8
009 W570285 GPO THA Lopinavir/Ritonavir NO 15 May 16 Positive 98.4/101.0 -2.53 1.94 96.8/99.9 99.8/102.7
010 W560556 GPO THA Lopinavir/Ritonavir NO 22 Oct 15 Positive 97.8/101.5 -1.47 1.70 99.1/101.4 101.7/103.7
011 W570169 GPO THA Lopinavir/Ritonavir NO 17 Mar 16 Positive 98.2/101.2 -1.33 1.52 94.9/100.0 97.6/102.8
012 8000458 Mylan IND Lopinavir/Ritonavir YES 30 Jun 16 Positive 99.7/101.4 -1.69 1.31 93.4/96.3 98.6/102.9

Abbreviations: Lopinavir,LPV; Ritonavir, RTV; the Government Pharmaceutical Organization, GPO; Thailand, THA; India, IND.