Table 5. Structure–Activity Relationships of Compounds Bearing Alkene Based Side Chains against SWI/SNF Bromodomainsa.


Values shown are the average of three replicates. Standard deviation is <0.6 °C. For PB1(3), values are a single measurement.


Values shown are the average of three replicates. Standard deviation is <0.6 °C. For PB1(3), values are a single measurement.