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. 2016 Feb 20;7(12):14616–14627. doi: 10.18632/oncotarget.7524

Table 1. Kinase profiling of Bakuchiol (20 μM).

Kinase Activity Kinase Activity Kinase Activity Kinase Activity Kinase Activity Kinase Activity
Abl 133 CDK9/cyclin T1 94 EGFR (T790M) 119 Lck 71 MST1 62 Rsk2 93
ASK1 68 CHK1 136 EGFR (T790M, L858R) 107 LKB1 85 mTOR 108 p38 51
Aurora-A 66 CHK2 97 FAK 100 Lyn 134 NEK7 102 SGK 151
Blk 47 CHK2 (I157T) 91 Fgr 98 MAPK1 78 p70S6K 172 SIK 108
CaMKI 85 CHK2 (R145W) 110 Flt1 93 MAPK2 113 PDK1 75 Src 95
CaMKIIβ 65 cKit 92 Fyn 102 MEK1 87 Pim-1 111 Syk 67
CDK1/cyclin B 84 CSK 147 GSK3β 49 Met 70 Pim-2 122 WNK2 82
CDK2/cyclin A 90 c-RAF 101 Hck 57 MKK4 108 Pim-3 80 Yes 134
CDK2/cyclin E 76 cSRC 87 IKKα 148 MKK6 94 PKA 120 ZAP-70 102
CDK3/cyclin E 100 DAPK1 80 JAK2 100 MKK7β 94 PKBα 109
CDK5/p25 94 DDR2 97 JAK3 79 MLK1 59 PKCα 109
CDK5/p35 111 EGFR 111 JNK1α1 98 Mnk2 84 Plk1 88
CDK6/cyclin D3 108 EGFR (L858R) 101 JNK2α2 100 MSK1 118 ROCK-I 84
CDK7/cyclin H 105 EGFR (L861Q) 105 KDR 92 MSK2 101 Rsk1 80