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. 2011 Jul 21;58(3):242–246. doi: 10.1016/S0377-1237(02)80139-3

TABLE 1.

Leukotrienes antagonists in asthma

Drug class Drug Usefulness Pediatric use
5-lipoxygenase inhibitor Zileuton Yes No
Cyst LT antagonist Montelukast Yes Yes
Pranlukast Yes No
Zafirlukast Yes Yes
FLAP antagonist BAY X 1005 No No
MK-886 No No
BLT antagonist LY-293111 No No