TABLE 1.
Leukotrienes antagonists in asthma
| Drug class | Drug | Usefulness | Pediatric use |
|---|---|---|---|
| 5-lipoxygenase inhibitor | Zileuton | Yes | No |
| Cyst LT antagonist | Montelukast | Yes | Yes |
| Pranlukast | Yes | No | |
| Zafirlukast | Yes | Yes | |
| FLAP antagonist | BAY X 1005 | No | No |
| MK-886 | No | No | |
| BLT antagonist | LY-293111 | No | No |