Table 5.

C3 analogs of ∆8-THC and ∆9-THC.

#		CB	NAME	CB1 KI (nM)	CB2 KI (nM)	FUNCTIONAL	REF
90		Δ8-THC		27.1 ± 4.5	51.5 ± 11.2	Agonist	100
91		Δ8-THC		0.3 ± 0.1	1.7 ± 0.4	Agonist	100
92		Δ8-THC		0.7 ± 0.2	3.0 ± 0.7	Agonist	100
93		Δ8-THC		0.8 ± 0.3	0.7 ± 0.2		99
94		Δ8-THC		0.5 ± 0.2	1.4 ± 0.7		99
95		Δ8-THC		3.4 ± 1.1	1.3 ± 0.3		99