Table 1.
Deletion constructs of LPHN3 and FLRT3 | ||||
---|---|---|---|---|
KD (nM) | LPHN3 | GAIN-HR | OLF-RBL | OLF |
FLRT3 | 31±7.9 | No binding | 43.3±13.8 | n.d. |
FN3 | No binding | n.d. | n.d. | n.d. |
LRR | n.d. | n.d. | 34.2±7.5 | 16.9±15.9 |
Amino-acid substitutions in LPHN3-OLF and FLRT3-LRR | ||||
---|---|---|---|---|
KD (nM) | LPHN3-OLF | LPHN3-OLF D332A | LPHN3-OLF Y323A | LPHN3-OLF A313S |
FLRT3-LRR | 17 | 170 | No binding | 19 |
FLRT3-LRR R117T | 27 | n.d. | n.d. | n.d. |
FLRT3-LRR F160N | No binding | n.d. | n.d. | n.d. |
FLRT3-LRR F160A | 1000 | n.d. | n.d. | n.d. |