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. Author manuscript; available in PMC: 2017 Aug 8.
Published in final edited form as: Eur J Med Chem. 2016 Apr 14;118:208–218. doi: 10.1016/j.ejmech.2016.04.033

Table 1.

IC50 value of the prepared amidine-functionalized analogs and the crystal ligand CA-14

Compound IC50 (μM)
13 23 ± 2.4
14 70 ± 6.4
15 44 ± 3.8
16 5.9 ± 0.5
17 11 ± 1.5
18 9.3 ± 0.4
19 8.9 ± 2.8
20 7.3 ± 0.3
21 14 ± 0.8
30 2.8 ± 0.9
CA-14 2.6 ± 0.1