Table 1.
Antimicrobial activity of γ-AApeptides.
Organism | MIC (µg/mL) | ||||
---|---|---|---|---|---|
γ-AA9 | γ-AA10 | γ-AA11 | γ-AA12 | γ-AA13 | |
Gram-negative | |||||
E. Coli | 5 | 3 | 4 | - | 2 |
P. aeruginosa | >50 | 3 | 4 | 8 | 5 |
Gram-Positive | |||||
MRSE | 5 | 3 | 2 | 2 | 1 |
E. faecalis | 5 | 4 | 2 | 5 | 3 |
MRSA | 5 | 3 | 2 | 1 | 2 |
Hemolysis (HC50) | 300 | >500 | >500 | 150 | 250 |