Table S1.
Kd values of bromodomains to BETi GS-626510
| Compound name | DiscoveRx gene symbol | Entrez gene symbol | Modifier | Kd (nM) |
| GS-626510 | ATAD2A | ATAD2 | > | 10,000 |
| GS-626510 | ATAD2B | ATAD2B | > | 10,000 |
| GS-626510 | BAZ2A | BAZ2A | > | 10,000 |
| GS-626510 | BAZ2B | BAZ2B | > | 10,000 |
| GS-626510 | BRD1 | BRD1 | > | 10,000 |
| GS-626510 | BRD2 (1) | BRD2 | = | 2.5 |
| GS-626510 | BRD2 (1, 2) | BRD2 | = | 1.1 |
| GS-626510 | BRD2 (2) | BRD2 | = | 0.59 |
| GS-626510 | BRD3 (1) | BRD3 | = | 1.7 |
| GS-626510 | BRD3 (1, 2) | BRD3 | = | 0.66 |
| GS-626510 | BRD3 (2) | BRD3 | = | 0.65 |
| GS-626510 | BRD4 (1) | BRD4 | = | 2.9 |
| GS-626510 | BRD4 (1, 2) | BRD4 | = | 1.3 |
| GS-626510 | BRD4 (2) | BRD4 | = | 3.2 |
| GS-626510 | BRD4 (full-length,short-iso.) | BRD4 | = | 2.8 |
| GS-626510 | BRD7 | BRD7 | > | 10,000 |
| GS-626510 | BRD8 (1) | BRD8 | = | 5,900 |
| GS-626510 | BRD8 (2) | BRD8 | > | 10,000 |
| GS-626510 | BRD9 | BRD9 | > | 10,000 |
| GS-626510 | BRDT (1) | BRDT | = | 19 |
| GS-626510 | BRDT (1, 2) | BRDT | = | 4.9 |
| GS-626510 | BRDT (2) | BRDT | = | 5 |
| GS-626510 | BRPF1 | BRPF1 | = | 4,100 |
| GS-626510 | BRPF3 | BRPF3 | > | 10,000 |
| GS-626510 | CECR2 | CECR2 | = | 8,200 |
| GS-626510 | CREBBP | CREBBP | = | 170 |
| GS-626510 | EP300 | EP300 | = | 220 |
| GS-626510 | FALZ | BPTF | > | 10,000 |
| GS-626510 | GCN5L2 | KAT2A | > | 10,000 |
| GS-626510 | PBRM1 (2) | PBRM1 | > | 10,000 |
| GS-626510 | PBRM1 (5) | PBRM1 | > | 10,000 |
| GS-626510 | PCAF | KAT2B | > | 10,000 |
| GS-626510 | SMARCA2 | SMARCA2 | > | 10,000 |
| GS-626510 | SMARCA4 | SMARCA4 | > | 10,000 |
| GS-626510 | TAF1 (2) | TAF1 | = | 8,000 |
| GS-626510 | TAF1L (2) | TAF1L | > | 10,000 |
| GS-626510 | TRIM24 (Bromo.) | TRIM24 | = | 4,100 |
| GS-626510 | TRIM24 (PHD, Bromo.) | TRIM24 | = | 6,900 |
| GS-626510 | TRIM33 (PHD, Bromo.) | TRIM33 | > | 10,000 |
| GS-626510 | WDR9 (2) | BRWD1 | > | 10,000 |