Table 2.
Summary for m708.5 in combination with drugs against neuroblastoma.
Drugs | LAN-1
|
SK-N-MM
|
||||||
---|---|---|---|---|---|---|---|---|
m708.5 | Drug | CIa ± SD | Effectb | m708.5 | Drug | CIa ± SD | Effectb | |
SN38 | 0.3μg/ml | 0.4–100nmol/L | 0.37 ± 0.05 | synergism | 0.6μg/ml | 0.4–100nmol/L | 0.48 ± 0.05 | synergism |
doxorubicin | 0.3μg/ml | 0.08–2μmol/L | 0.52 ± 0.03 | synergism | 0.6μg/ml | 0.08–2μmol/L | 0.61 ± 0.12 | synergism |
vincristine | 0.3μg/ml | 0.2–60nmol/L | 0.6 ± 0.19 | synergism | 0.6μg/ml | 0.2–60 | 0.59 ± 0.02 | synergism |
cisplatin | 0.3μg/ml | 0.4–100μmol/L | 0.80 ± 0.00 | moderate synergism | 0.6v | 0.4–100μmol/L | 1.28 ± 0.07 | moderate antagonism |
temsirolimus | 0.3μg/ml | 0.2–5μmol/L | 0.49 ± 0.28 | synergism | 0.6μg/ml | 0.2–5μmol/L | 0.18 ± 0.04 | strong synergism |
CI, combination index
definition of CI values, <0.1(very strong synergism); 0.1–0.3 (strong synergism); 0.3–0.7 (synergism); 0.7–0.85 (modest synergism); 0.85–0.9 (slight synergism); 0.9–1.1 (nearly additive); 1.1–1.2 (slight antagonism); 1.2–1.45 (modest antagonism); 1.45–3.3 (antagonism);3.3–10 (strong antagonism); >10 (very strong antagonism).