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. 2016 Aug 10;7:248. doi: 10.3389/fphar.2016.00248

Table 3.

Tabular summary of the medicinal plants used by the patients and their pharmacokinetic profile.

Botanical name of medicinal plant (Common/Local name as used by patient) Number of Patients (%) Effect on intestinal P-gp or other absorption mechanisms Effect on cytochromes or other hepatic enzymes (GSTs, ALT, AST) Other toxic effects
Vernonia amygdalina Delile (Bitter leaf/Onugbu) 13 (11.6) Inhibits P-gp efflux activity (Oga et al., 2012)
Ocimum gratissimum L. (Scent leaf/Nchonwu) 5 (4.5) Dose dependent increase in AST and ALT levels (Ajibade et al., 2012)
Musa paradisiaca (Plantain/Banana) 3 (2.7) Polyvalent cations in the plant form non-absorbable complexes with certain drugs (Nwafor et al., 2003)
Mangifera indica L. (Mango) 3 (2.7) Inhibits the P-gp efflux activity (Chieli et al., 2009) Inhibits CYP 1A1/2 and 3A4 activities in rat liver microsomes (Rodeiro et al., 2009)
Persea americana Mill. (Avocado pear) 2 (1.8) Inhibits CYP 3A4/5/7 enzymes to different extents (Agbonon et al., 2010)
Gongronema latifolium Benth. (Utazi) 1 (0.9)
Abelmoschus esculentus (L.) Moench (Okro) 1 (0.9) Water soluble fractions inhibits metformin absorption in vivo (Khatun et al., 2011)
Anarcadium occidentale L. (Cashew) 1 (0.9)
Azadirachta indica A. Juss. (Neem) 1 (0.9) Pharmacotoxic effects of neem oil in lungs and CNS (Gandhi et al., 1988)
Camellia sinensis (L.) Kuntze (Tea) 1 (0.9)
Picralima nitida (Stapf) T. Durand and H. Durand (Mkpokiri/Abere) 1 (0.9) Elevated AST, ALT, and GSH levels (Kouitcheu Mabeku et al., 2008) Hepatotoxic effects (Fakeye et al., 2004)
Terminalia catappa L. (Tropical almond) 1 (0.9) Hepatotoxic at high doses due to punicalagin (Lin et al., 2001)
Unknown 36 (31.9) NA NA NA
Discontinued 14 (12.4) NA NA NA