Skip to main content
. 2016 Jun 1;7(8):735–740. doi: 10.1021/acsmedchemlett.6b00167

Table 2. Pharmacokinetic Parameters of 12 in Male Sprague Dawley Rats Following IV and PO Dosing.

  1 mg/kg iva 15 mg/kg pob
Cl [mL/min/kg] 84 NA
Vd [L/kg] 10 NA
t1/2 [h] 1.7 NA
AUC0-inf [nM·h] 396 2370
Cmax [nM] NA 225
BAV [%] NA 40
a

NMP/PEG200 (30:70).

b

MEPC5/Water (10:90).