Skip to main content
. 2016 Aug 17;6:31633. doi: 10.1038/srep31633

Table 5. Antiproliferative activities of some compounds from T. chinensis against human cancer cell lines.

Compound IC50 (μM)a
FaDu Detroit 562 CNE-1 CNE-2 HepG2 K562 SPC-A-1
3 28.6 ± 1.6* >50.0 >50.0 >50.0 >50.0 >50.0 >50.0
4 27.6 ± 3.6*** >50.0 >50.0 >50.0 29.7 ± 3.1*** >50.0 >50.0
5 41.2 ± 1.8*** >50.0 >50.0 >50.0 >50.0 >50.0 >50.0
12 12.1 ± 1.2 >50.0 >50.0 >50.0 >50.0 >50.0 >50.0
17 20.3 ± 2.1 20.2 ± 2.0 33.6 ± 0.3*** 23.6 ± 1.9*** 28.6 ± 1.0*** 27.4 ± 0.2*** 24.8 ± 0.7***
18 >50.0 39.4 ± 0.7*** >50.0 40.7 ± 3.1*** 46.5 ± 1.0*** >50.0 >50.0
19 61.4 ± 2.5*** 21.5 ± 1.1*** 50.9 ± 1.1*** 29.5 ± 0.9*** 34.0 ± 0.5*** 40.2 ± 2.1*** 39.4 ± 1.0***
20 20.1 ± 0.4 20.1 ± 0.6*** >50.0 >50.0 28.0 ± 0.7*** >50.0 >50.0
21 12.7 ± 1.7* 22.7 ± 0.5** 17.4 ± 0.5*** 14.5 ± 1.1** 14.3 ± 1.5*** 22.2 ± 0.2*** 22.2 ± 0.2***
22 20.5 ± 3.4 29.1 ± 0.6* 33.7 ± 0.6*** >50.0 17.7 ± 0.3*** 33.8 ± 0.1*** 26.3 ± 1.0***
CISb 18.1 ± 0.7 26.2 ± 1.5 10.8 ± 0.4 7.9 ± 1.1 6.5 ± 0.3 13.5 ± 0.8 3.8 ± 0.3

aValues are presented as means ± SD (n = 3).

bPositive control.

*p < 0.05, **p < 0.01, ***p < 0.001 versus positive control.