TARGETS
GPCRs a
5‐HT2C receptor
β2‐adrenoceptor
A2A adenosine receptor
GPR50
MT1 receptor
MT2 receptor
Voltage‐gated ion channels b
Cav2.2 channels
Transporters c
GLUT1
Enzymes d
CaMKII
ERK1

LIGANDS
6‐Chloromelatonin	CIFEA	[3H]‐melatonin
5‐HEAT	Difluoroagomelatine	Ramelteon
6‐Hydroxymelatonin	[125I]‐DIV880	S22153
2‐(indolin‐1yl)‐melatonin	Dopamine	S24014
2‐Iodomelatonin	EFPPEA	S24773
2‐[125I]iodomelatonin	fMLP	S26131
2‐Methoxy‐α,β‐didehydro‐agomelatine	GR 128107	S26284
5‐Methoxyluzindole	GR 196429	Tasimelteon
4P‐PDOT	(Hydroxymethylphenyl) agomelatine	TNF
[125I]‐SD6	IIK7	TIK 301
[125I]‐S70254	isoamyl agomelatine	UCM 454
AAE‐M‐PBP amine	K185	UCM 765
Agomelatine	Luzindole	UCM 793
BOMPPA	MCA‐NAT	UCM1014
cAMP	N‐acetyl‐serotonin
CBOBNEA	Melatonin

These Tables list key protein targets and ligands in this article which are hyperlinked to corresponding entries in http://www.guidetopharmacology.org, the common portal for data from the IUPHAR/BPS Guide to PHARMACOLOGY (Southan et al., 2016) and are permanently archived in the Concise Guide to PHARMACOLOGY 2015/16 (^a,b,c,dAlexander et al., 2015a, 2015b, 2015c, 2015d).