Table 3.
IC50 and Hill coefficient for the different CaV1.2 splice variants. IC50 and Hill coefficient (h) from fits of data as in Fig. 2 with the equation I (concentration) = I(0) ∗ 1 / (1 + (IC50 / [concentration])h).
Clones | Drug | IC50 (μM) | h |
---|---|---|---|
22-32-33 | Clevidipine | 0.22 | 0.85 |
22-32-33 | Nicardipine | 2.01 | 0.85 |
21-31-33 | Clevidipine | 0.19 | 0.82 |
22-31-delta33 | Clevidipine | 0.06 | 0.8 |
22-31-delta33 | Nicardipine | 0.885 | 1.03 |
22-32-delta33 | Clevidipine | 0.19 | 1.1 |
21-32-delta33 | Clevidipine | 0.28 | 1.04 |
21-31-delta33 | Clevidipine | 0.16 | 0.9 |