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. 2016 Jun 22;10:291–297. doi: 10.1016/j.ebiom.2016.06.027

Table 3.

IC50 and Hill coefficient for the different CaV1.2 splice variants. IC50 and Hill coefficient (h) from fits of data as in Fig. 2 with the equation I (concentration) = I(0) ∗ 1 / (1 + (IC50 / [concentration])h).

Clones Drug IC50 (μM) h
22-32-33 Clevidipine 0.22 0.85
22-32-33 Nicardipine 2.01 0.85
21-31-33 Clevidipine 0.19 0.82
22-31-delta33 Clevidipine 0.06 0.8
22-31-delta33 Nicardipine 0.885 1.03
22-32-delta33 Clevidipine 0.19 1.1
21-32-delta33 Clevidipine 0.28 1.04
21-31-delta33 Clevidipine 0.16 0.9