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. 2016 Mar 1;7(16):21658–21675. doi: 10.18632/oncotarget.7808

Table 1. EC50a (μM) derived from TO displacement (FID) by selected AQ and AN derivatives from G4 folded KIT sequences.

AQ1 AQ5 AQ3 AQ7 AN6
KIT1 0.32 ± 0.05 0.27 ± 0.02 0.50 ± 0.04 0.24 ± 0.04 4.11 ± 0.70
KIT2 0.35 ± 0.05 0.41 ± 0.03 0.62 ± 0.05 0.25 ± 0.02 3.63 ± 1.00
a

ligand concentration that displaces 50% of TO from tested DNA sequences.