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. 2016 Sep 14;11(9):e0162594. doi: 10.1371/journal.pone.0162594

Table 2. ARQ 087 GI50 in Ba/F3 transfected cell lines.

Kinase GI50 (nM) Kinase GI50 (nM)
FGFR3-BAIAP2L1 34.9 FGFR2-CCD6 1121
FGFR2-CIT 39.5 FYN 1329
TEL-FGFR2 59.8 FGFR3 1337
FGFR2 232 FGFR4 1346
ARG 247 FLT4 (VEGFR3) 1354
LCK 287 LYN 1363
FGFR2-AFF3 337 PDFGR-β 1376
FGFR2-CASP7 349 FLT1 (VGFR1) 1407
FGFR1 355 PDFGFR-α 1567
KIT 474 IGF1R 1546
FGFR2-BICC1 990 KDR (VEGFR2) 1557
RET 991 FMS 1710
SRC 1091 EphA1 5381