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. Author manuscript; available in PMC: 2017 May 26.
Published in final edited form as: J Med Chem. 2016 May 3;59(10):4800–4811. doi: 10.1021/acs.jmedchem.6b00012

Figure 1.

Figure 1

Fragment hit 1, a commercially sourced screening hit 2 and a novel, chemically synthesized analogue 3 with representative DSF data at 10 μM against the PB1(5) bromodomain.