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CDK9 Inhibition K1 values by small molecules 1–10. 
| Number | Name | Inhibition K1 (nM) |
|---|---|---|
| 1 | Flavopiridol39 | 4.59 |
| 2 | CR837,53 | 110 |
| 3 | Indirubin-3´-monoxime derivatives38 | 400 |
| 4 | 5-Fluoro-N2,N4-diphenylpyrimidine-2,4-diamines39 | 330 |
| 5 | 4-(thiazol-5-yl)-2-(phenylamino)pyrimidines40,50 | 7 |
| 6 | TG0248,49,54 | 3 |
| 7 | CDKI-7348 | 4 |
| 8 | 2,4,5-trisubstited pyrimidine derivatives49 | 14 |
| 9 | LCD00006751 | 44 |
| 10 | Wogonin52 | 190 |
