Table 1.
Pharmacokinetics of orally delivered Taxotere® and enteric microparticles containing docetaxel PLGA nanocaspules (both equivalent to 1.25 mg/kg of docetaxel) in minipigs (n=3). Enteric microparticles containing docetaxel PLGA nanocaspules showed significantly higher Cmax and AUC as compared to Taxotere® (p < 0.05). Adapted from reference [193] with permission
Oral Formulation | Cmax (ng/mL) | AUC (h.ng/mL) | Clearance (L/h/kg) |
---|---|---|---|
Docetaxel solution | 97.6 ± 221 | 797.7 ± 1141 | 4 ± 2.8 |
Enteric microparticles containing docetaxel PLGA nanocaspules | 827.9 ± 558 | 7923.1 ± 5644 | 0.4 ± 0.5 |