Table 1. Search result of query "imatinib resistance ABL1" with type filter "mutations.".
Rank | BEST result | BEST score | ABL1 mutation | Known Imatinib binding site in ABL1 [10,11] | Acquired mutations found in CML patient resistant to imatinib |
---|---|---|---|---|---|
1 | T315I | 24.520 | Yes | Yes | Yes |
2 | Y253H | 7.744 | Yes | Yes | Yes |
3 | E255K | 5.602 | Yes | Yes | |
4 | E355G | 2.871 | Yes | Yes | |
5 | G250E | 2.757 | Yes | Yes | |
6 | G398R | 2.048 | Yes | Yes | |
7 | M351T | 1.430 | Yes | Yes | |
8 | Q252H | 1.349 | Yes | Yes | |
9 | E255V | 1.328 | Yes | Yes | |
10 | V289F | 1.218 | Yes | Yes | Yes |