Table 2.
siRNA | siINDY* (unmodified) | siINDY |
---|---|---|
IC50KD (nM) | 0.15 | 0.56 |
ImaxKD (%) | 92 | 92 |
Serum stability (h): t1/2 in 50% mouse serum | <2 | 4 |
Cytotoxicity (%): Viability of Hepa1c1c7 cells | 78 | 135 |
Immune stimulation (pg/ml): IFNα release PBMCs | 2144 | 70 |
ImaxKD: maximal knockdown of mINDY mRNA expression.