Table 3.
Effect of Constrained pTyr Surrogates on the Affinity of Xaa-Lys-Pro-Phe-NH2
| Xaa | IC50(µM) | ||
|---|---|---|---|
| 5 | Ac-pTyr |  |
6.1 ± 1.2 |
| 14 | pCinn |  |
8.6 ± 2.8 |
| 15 | p-Indole |  |
3.7 ± 0.052 |
| 16 | p-Benzofuran |  |
89.6 ± 1.5 |
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