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. Author manuscript; available in PMC: 2016 Nov 15.
Published in final edited form as: J Med Chem. 2015 Nov 9;58(22):8970–8984. doi: 10.1021/acs.jmedchem.5b01321

Table 6.

Effect of Proline Replacements on βMpCinn-Tle-Xaa-N(Me)Ph

Xaa IC50 (µM)
19c proline 0.12 ± 0.03
21 sarcosine 0.27 ± 0.05
22 alanine 0.12 ± 0.016
23 N-methyl-alanine 0.48 ± 0.094