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. 2016 Sep 28;291(47):24628–24640. doi: 10.1074/jbc.M116.738567

TABLE 4.

Metabolic stability of ML364

Rat microsomal stability, t½a Mouse microsomal stability, (remaining at 30 min)b Human microsomal stability, (remaining at 30 min)b Mouse plasma stability (remaining at 30 min)a
ML364 15 min 61% 84% 100%

a Performed in-house.

b Contracted to Pharmaron, Inc.