Table 1.
Kon (M−1s−1) | Koff (s−1) | KD (M) | KD wt / KD Matured | |||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|
1aE2 | F442I E2 | F442L E2 | 1aE2 | F442I E2 | F442L E2 | 1aE2 | F442I E2 | F442L E2 | 1aE2 | F442I E2 | F442L E2 | |
HC84.26 | 1.3E+04 | 3.2E+03 | 5.6E+03 | 2.1E−04 | 6.3E−03 | 1.6E−03 | 1.6E−08 | 2.0E−06 | 2.8E−07 | 1.0 | 1.0 | 1.0 |
HC84.26.5 | 3.2E+04 | 1.3E+04 | 1.2E+04 | 2.5E−04 | 1.7E−03 | 1.1E−03 | 7.7E−09 | 1.3E−07 | 8.9E−08 | 2.1 | 15.7 | 3.2 |
HC84.26.5D | 2.0E+04 | 1.1E+04 | 9.7E+03 | 1.3E−04 | 6.5E−04 | 4.4E−04 | 6.4E−09 | 5.8E−08 | 4.5E−08 | 2.5 | 34.0 | 6.3 |
HC84.26.5G | 2.3E+04 | 1.3E+04 | 1.1E+04 | 8.5E−05 | 9.7E−04 | 6.7E−04 | 3.6E−09 | 7.7E−08 | 5.9E−08 | 4.4 | 26.0 | 4.8 |
HC84.26.5DG | 2.7E+04 | 1.1E+04 | 1.0E+04 | 1.7E−04 | 8.7E−04 | 5.1E−04 | 6.3E−09 | 8.0E−08 | 4.9E−08 | 2.5 | 25.0 | 5.8 |