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. 2016 Sep 15;7(12):1028–1033. doi: 10.1021/acsmedchemlett.6b00184

Table 5. Inhibitory Activity toward DHT-Promoted SC-3 Cell Proliferation.

compd inhibition at 1 μM (%)a
7 66 ± 2.1
20a 8.4 ± 23
29 N.D.b
30 N.D.b
32 N.D.b
a

Cell proliferation was promoted by 1 nM DHT.

b

No inhibition was observed.