| Berkazaphilone A (25): | IC100 | Caspase-1: 100 μg/mL |
| Berkazaphilone B (26): | IC100 | Caspase-1: 10 μg/mL |
| leukemia RPMI-8226: log10 GI50 (−5.67) | ||
| Berkazaphilone C (27): | IC100 | Caspase-1: 10 μg/mL |
| leukemia SR: log10 GI50 (−6.42) | ||
| Penisimplicissimum (30): | IC100 | Caspase-1: 100 μg/mL |
| leukemia CCRFCEM: log10 GI50 (−6.70) | ||
| leukemia HL-60: log10 GI50 (−5.83) | ||