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. Author manuscript; available in PMC: 2016 Dec 22.
Published in final edited form as: ChemMedChem. 2011 Sep 8;6(11):1961–1966. doi: 10.1002/cmdc.201100346

Figure 4.

Figure 4

Inhibition of APH(3′)-IIIa-catalyzed amikacin phosphorylation by analogue 20 as a function of ATP concentration. v=phosphorylation rates, ◆ =0 μM, × =1 μM, ▲=2.5 μM, ●=5 μM, ■=10 μM.