Table 2.
Constants
R0 | Total receptor concentration (nM) |
GQ0 | Total Gq/11 protein concentration (nM) |
ERUL | Resting Ca2+ concentration in ER (normally 40 μM) |
CAE | External Ca2+ concentration (normally 1000 μM) |
α | = 2 nM-1, see equation (17) |
β | = 4 min-1, see equation (17) |
v1 | = 0.02 min-1, see equation (12) |
v2 | = 0.002 min-1, see equation (12) |
r0 | = 0.6, fraction internalized receptors returned |
P0 | = 8.3 × 10-6 nM·min-1, basal rate of receptor synthesis |
γ | = 8.3 × 10-4 min-1, basal rate of receptor degradation |
k1 | = 2.5 nM-1·min-1 |
k-1 | = 5 min-1 |
k2 | = 2500 nM-1·min-1 |
k-2 | = 5 min-1 |
k3 | = 4000 nM-1·min-1 |
k-3 | = 200 min-1 |
k5 | = 2 × 107 min-1 |
k-5 | = 10 min-1 |
k6 | = 1 nM-1·min-1 |
k66 | = 10 nM-1·min-1 |
k666 | = 0 |
k-6 | = 5 min-1 |
k7 | = 2.2 μM·min-1 |
k8 | = 0.4 nM-1·min-1 |
k88 | = 0 |
k888 | = 0 |
k9 | = 0.0002 min-1 |
k10 | = 5 ng·min-1 |
k11 | = 0.0008 nM-1·min-1 |
k33 | = 2.7 min-1 |