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. Author manuscript; available in PMC: 2017 Dec 1.
Published in final edited form as: Pharm Res. 2016 Aug 15;33(12):2930–2942. doi: 10.1007/s11095-016-2015-0

Table 1.

Unidirectional drug uptake into brain transfer constant (Kin) values. Results are presented as Mean ± STDEV

Test article Kin
(mL/s/g)
BDTa area Number Tumor area Number
BTA (1.68±0.33)×10−7 61 (11.01±7.21)×10−7 336
hMTf (p97) (1.84±0.38)×10−5 49 (5.30±3.97)×10−5 167
BT2111 (2.31±0.60)×10−6 52 (11.70±8.29)×10−6 101
(7.32±2.41)×10−6 24 (9.88±3.44)×10−6 112
(3.89±2.71)×10−6 76 (10.74±6.28)×10−6 213
a

Brain Distant to Tumor (normal brain, BDT) area