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Overview of PI3K inhibitors
| Class | Substance |
|---|---|
| Pan-PI3K inhibitors | BKM120 (buparlisib) |
| XL-147 | |
| PX-866 | |
| PKI-587 | |
| GDC-0941 | |
| p110α-specific inhibitors | wortmannin |
| LY294002 | |
| BYL719 (alpelisib) | |
| GDC-0032 | |
| INK-1117 | |
| p110δ-specific inhibitors | CAL-101 |
| Dual PI3K/mTOR inhibitors | BEZ235 |
| BGT226 | |
| PF-4691502 | |
| GDC-0980 | |
| XL-765 |
