Table 4. Androgen receptor splice variants.
Variant | Protein Regions | Activity | References |
---|---|---|---|
ARV7 (AR3) | NTD, DBD | Ligand-independent, Nuclear | [119–120,122–123, 126] |
ARv567es | NTD, DBD, Hinge | Ligand-independent, Nuclear | [121, 126] |
ARV12 | NTD, DBD, Hinge | Ligand-independent, Nuclear | [123] |
AR1/2/2b (ARV3) | NTD, partial DBD | Ligand-independent | [118–120] |
AR1/2/3/2b (ARV4, AR5) | NTD, DBD | Ligand-independent | [118–120] |
ARV1 (AR4) | NTD, DBD | LNCaP: Ligand-independent, PC3: Inactive, Cytoplasmic | [119–120, 123,126] |
ARV9 | NTD, DBD | LNCaP: Ligand-independent, PC3: Inactive, Cytoplasmic | [123, 126] |
ARV13 | NTD, DBD, Hinge, partial LBD | Inactive | [123] |
ARV2 | NTD, DBD | Not determined | [119] |
ARV5/V6 | NTD, DBD | Not determined | [119] |
ARV8/10/11 | NTD, DBD | Not determined | [126] |
ARV14 | NTD, DBD, Hinge, partial LBD | Not determined | [123] |