TABLE 4.
Study size and dosingb | % AUC0t | % AUCinf | % Cmax | % Tmax | % BE0t | % BEinf |
---|---|---|---|---|---|---|
12 participants per study | ||||||
Doryx MPC vs Doryx tablet (Fasted) | 89.8 | 87.9 | 88.1 | 15.7 | 79.2 | 77.8 |
Doryx MPC vs Doryx tablet (Fed) | 90.5 | 86.7 | 7.5 | 0 | 6 | 5.6 |
Doryx MPC vs Doryx MPC (Fed/Fasted) | 62.4 | 60.5 | 0 | 0 | 0 | 0 |
Doryx tablet vs Doryx tablet (Fed/Fasted) | 65.2 | 61.1 | 12.2 | 5 | 8.6 | 8.1 |
24 participants per study (1,000 simulated studies) | ||||||
Doryx MPC vs Doryx tablet (Fasted) | 99.7 | 99.6 | 99.8 | 58.6 | 99.5 | 99.4 |
Doryx MPC vs Doryx tablet (Fed) | 99.6 | 99.5 | 7.6 | 0 | 7.4 | 7.3 |
Doryx MPC vs Doryx MPC (Fed/Fasted) | 88 | 85.9 | 0 | 0 | 0 | 0 |
Doryx tablet vs Doryx tablet (Fed/Fasted) | 88.4 | 86 | 18.4 | 6.3 | 16.8 | 16.3 |
28 participants per study | ||||||
Doryx MPC vs Doryx tablet (Fasted) | 99.8 | 99.7 | 99.8 | 67.4 | 99.6 | 99.5 |
Doryx MPC vs Doryx tablet (Fed) | 99.8 | 99.6 | 8.9 | 0 | 8.8 | 8.7 |
Doryx MPC vs Doryx MPC (Fed/Fasted) | 92 | 90.6 | 0 | 0 | 0 | 0 |
Doryx tablet vs Doryx tablet (Fed/Fasted) | 93.6 | 91.2 | 19 | 4.7 | 17.8 | 17.7 |
36 participants per study | ||||||
Doryx MPC vs Doryx tablet (Fasted) | 100 | 100 | 100 | 82 | 100 | 100 |
Doryx MPC vs Doryx tablet (Fed) | 100 | 100 | 9.1 | 0 | 9.1 | 9.1 |
Doryx MPC vs Doryx MPC (Fed/Fasted) | 95.8 | 95.1 | 0 | 0 | 0 | 0 |
Doryx tablet vs Doryx tablet (Fed/Fasted) | 96.4 | 95.3 | 21.2 | 5.8 | 20.8 | 20.7 |
Percent AUCinf, AUC0t, Cmax, and Tmax indicates, respectively, the power percentage for a study to display equivalence of AUCinf, AUC0t, Cmax, and Tmax for the crossover designs indicated. Percent BE0t and BEinf indicates, respectively, the power percentage for a study to display bioequivalence via AUC0t and Cmax and via AUCinf and Cmax for the crossover designs indicated.
For the studies, 120 mg of Doryx MPC and 100-mg Doryx tablets were used. For each group, 1,000 simulated studies were performed.