Table 1. Drugs used in screen.
Drug | Target | Libraries screened |
---|---|---|
Camptothecin | Topoisomerase I | 1, 6, 7, 8, 9, 10 |
BIIB021 | HSP90 | 1, 2, 3, 6, 7, 8, 9, 10, 2sims |
AT13387 | HSP90 | 1, 6, 7, 8, 9, 10 |
Bleomycin | Double strand breaks | 1, 6, 7, 8, 10 |
Methotrexate | DHFR | 1, 2, 3, 7, 8, 9, 10, 2sims |
JQ1 | BRD4 | 1, 2, 3, 4, 6, 7, 8, 9, 2sims |
KW2478 | HSP90 | 1, 6, 7, 9, 10 |
BMN 673 | PARP1/2 | 1, 2, 3, 4, 6, 7, 8, 10, 2sims |
MK1775 | WEE1 | 1 |
17-AAG | HSP90 | 1, 7, 8, 9, 10 |
Etoposide | Topoisomerase II | 1, 6, 7, 10 |
Decitabine | DNA methyltransferase | 1, 6, 7, 8, 9, 10 |
PF04691502 | HSP90 | 1, 8, 9, 10 |