Table 1.
Receptor | pKi* | n** | Radioligand |
A2A | 7.95 ± 0.06 | 4 | [3H]-ZM241385 |
A1 | 6.8 | 2 | [3H]-DPCPX |
NR2B | 8.25 ± 0.17 | 4 | [3H]-UCB9352*** |
Negative logarithm of the equilibrium dissociation constant of Cmpd-1 determined by competitive binding assay.
Number of parallel tests for the binding assay.
Proprietary compound of UCB.