TARGETS
GPCRs a					Enzymes b
5‐HT1B receptor	GPR4	GPR32	GPR78	MRGPRD	AC
5‐HT2B receptor	GPR6	GPR34	GPR82	MRGPRE	ERK1
α1A‐adrenoceptor	GPR10	GPR35	GPR83	MRGPRF	ERK2
β1‐adrenoceptor	GPR11	GPR37	GPR84	MRGPRG	MAPK
β2‐adrenoceptor	GPR12	GPR37L1	GPR85	MRGPRX1	MEK
δ receptor	GPR13	GPR39	GPR87	MRGPRX2	MEKK
κ receptor	GPR14	GPR40	GPR88	MRGPRX4	PKC
A2A receptor	GPR15	GPR43	GPR92	MT1 receptor	PLC
AT1 receptor	GPR16	GPR45	GPR97	NOP receptor	Raf
BB3 receptor	GPR17	GPR50	GPR99	OPN3	Ste7
CXCR4	GPR18	GPR51	GPR139	OPN4	Ste11
CXCR7 (ACKR3)	GPR19	GPR52	H1 receptor	OPN5
D2 receptor	GPR20	GPR55	H4 receptor	P2Y1 receptor
D3 receptor	GPR21	GPR61	LGR4	P2RY8
FFA1 receptor	GPR22	GPR62	LGR5	TAAR2
FFA2 receptor	GPR25	GPR63	LGR6	TAAR5
FFA3 receptor	GPR26	GPR65	M3 receptor	TAAR6
GPR1	GPR27	GPR68	MAS1	TAAR8
GPR3	GPR31	GPR75	MAS1L	TAAR9

LIGANDS
Acetate
ATP
cAMP
GW9508
IP3
Linoleic acid
Nateglinide
TAK‐875