Skip to main content
. Author manuscript; available in PMC: 2017 Mar 10.
Published in final edited form as: Prog Chem Org Nat Prod. 2017;103:103–131. doi: 10.1007/978-3-319-45541-9_4

Table 3.

Activation of PPAR isotypes by phytocannabinoids.

pCBs PPARα PPARβ/δ PPARγ
Δ9-THC Transcriptional
activity [104]
- Binding assays [106]
Transcriptional activity [105]
Inhibition by PPARγ antagonists [19, 105]
CBD - - Binding assays [106]
Transcriptional activity [47]
Inhibition by PPARγ antagonists[4749]
CBG - - Binding assays [106]
CBC - - Binding assays [106]
THCV - - NR [18]

NR: No response