Table 1. In Vitro Inhibitory Activities of Compounds 7a–7j against DDR1, DRR2, Bcl-Abl, and c-Kita.
DDR1 and DDR2 experiments were performed using LANCE ULTRA kinase assay according to the manufacturer’s instructions. Bcr-Abl and c-Kit activity experiments were performed using the förster resonance energy transfer (FRET)-based Z′-Lyte assay according to the manufacturer’s instructions. All the data are mean values from at least three independent experiments.