Table 4.
Three-Parameter QSRR Model | ||||||||
---|---|---|---|---|---|---|---|---|
EVO | Gemini | |||||||
MDs | G1 | G2 | G3 | G4 | G1 | G2 | G3 | G4 |
pKa1 | −0.82 ± 0.30 | −0.60 ± 0.32 | −0.61 ± 0.24 | −0.41 ± 0.50 | −1.08 ± 0.30 | −0.74 ± 0.37 | −0.71 ± 0.15 | −0.56 ± 0.65 |
pKa2 | 1.17 ± 0.13 | 0.86 ± 0.14 | 1.01 ± 0.11 | 0.73 ± 0.22 | 1.52 ± 0.13 | 1.09 ± 0.18 | 1.27 ± 0.07 | 0.93 ± 0.29 |
logP | 2.30 ± 0.57 | 1.96 ± 0.62 | 1.63 ± 0.47 | 2.36 ± 0.96 | 2.91 ± 0.58 | 2.04 ± 0.76 | 2.24 ± 0.29 | 2.22 ± 1.05 |
1.2/2.8/1.9 1 | 1.3/3.1/2.1 1 | 1.0/2.4/1.6 1 | 1.8/5.8/3.2 1 | 1.1/2.9/1.9 1 | 1.6/3.6/2.5 1 | 0.6/1.4/1.0 1 | 2.5/6.9/4.2 1 |
1 Average absolute difference of experimental and calculated tR/Maximum absolute difference of experimental and calculated tR/Standard error of the estimate SEE.