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. 2017 Apr 13;45(2):571–582. doi: 10.1042/BST20160182

Table 1. Iminosugar IC50 values against purified rat α-glucosidase I and II; experiments were performed using a Glc1-3Man7GlcNAc2 substrate.

Iminosugar α-glu I α-glu II
Glc2 Glc1
NB-DNJ 0.68 ± 0.05 10.80 ± 05 53.00 ± 6.6
NN-DNJ 0.54 ± 0.08 2.10 ± 0.42 14.90 ± 3.6
MON-DNJ 0.015 ± 0.04 0.90 ± 0.19 1.60 ± 0.2
NAP-DNJ 0.017 ± 0.01 0.30 ± 0.1 0.83 ± 0.13