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. 2017 Mar 9;8(4):413–417. doi: 10.1021/acsmedchemlett.6b00496

Table 1. Optimization of 10.

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a

Utilizing MOLT-4 (human T cell leukemia) cellular lysate, a proteasome constitutive/immunoproteasome subunit ELISA (ProCISE) was employed for quantitative assessment of subunit-specific activity. Data are reported as the mean ± SD (n ≥ 2).

b

Liver S9 data collected at 90 min without NADPH present. Data are reported as the mean ± SD (n ≥ 3).

c

Solubility data collected at pH 7.2. Data are reported as the mean ± SD (n = 2).