Table 2.
HIF Inhibition by Class 1A analogs
| ||
|---|---|---|
| Name | R1 | IC50[a] |
| 3a |
|
0.98 |
| 3b |
|
3.3 |
| 3c |
|
3.2 |
| 3d |
|
3.1 |
| 3e |
|
1.8 |
| 3f |
|
>5 |
| 3g |
|
>5 |
[a]
IC50 values are in micromolar (μM).
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