Table 5.
HIF Inhibition by Class 2A analogs
| ||
|---|---|---|
| Name | R1 | IC50[a] |
| 6a |
|
>5 |
| 6b |
|
3.9 |
| 6c |
|
>5 |
| 6d |
|
>5 |
| 6e |
|
>5 |
| 6f |
|
>5 |
| 6g |
|
1.0 |
| 6h |
|
1.3 |
| 6i |
|
3.5 |
[a]
IC50 values are in micromolar (μM).
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