Figure 4. Optimization of domino and one-pot processes.
(a) Four-component (ABC2) five-step branched domino reaction. (b,c) Optimization of one-pot two-step synthesis of 2,6-dicyanoaniline derivative 5a (see Supplementary Methods).
(a) Four-component (ABC2) five-step branched domino reaction. (b,c) Optimization of one-pot two-step synthesis of 2,6-dicyanoaniline derivative 5a (see Supplementary Methods).