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. Author manuscript; available in PMC: 2017 Jun 1.
Published in final edited form as: J Med Chem. 2017 Jan 31;60(3):1210–1218. doi: 10.1021/acs.jmedchem.6b01792

Figure 1.

Figure 1

Structure–activity analysis of aminophenyl-1,3,5-triazine CFTR activators. (A) Chemical structure of 1. (B) Preliminary SAR analysis based on commercial analogs (see Supporting Information Table 1 for data on all commercial analogs).