TABLE 4.
Effects of Pma1 inhibitors on Hep-G2 cells
| Compound | EC50 (μM) for Hep-G2 cells at 24 h |
|---|---|
| 14 | 2.3 ± 0.0 |
| 15 | 2.8 ± 0.1 |
| 16 | 2.6 ± 0.9 |
| 17 | 5.8 ± 1.1 |
| 18 | 3.6 ± 1.1 |
| 19 | 24.2 ± 0.5 |
| BM2 | >100 |
| Vanadate | >500 |
| Ebselen | 10.7 ± 7.0 |
Effects of Pma1 inhibitors on Hep-G2 cells
| Compound | EC50 (μM) for Hep-G2 cells at 24 h |
|---|---|
| 14 | 2.3 ± 0.0 |
| 15 | 2.8 ± 0.1 |
| 16 | 2.6 ± 0.9 |
| 17 | 5.8 ± 1.1 |
| 18 | 3.6 ± 1.1 |
| 19 | 24.2 ± 0.5 |
| BM2 | >100 |
| Vanadate | >500 |
| Ebselen | 10.7 ± 7.0 |