Table 1.
Radioactivity in liver, kidney and blood/tissue ratios via QWBA
| WT | 6 h | 24 h | 72 h | |||
|---|---|---|---|---|---|---|
| dpm/g | Tissue/blood | dpm/g | Tissue/blood | dpm/g | Tissue/blood | |
| Blood | 3150,670 | 1.00 | 1266,494 | 1.00 | 145,195 | 1.00 |
| Brain | 81,217 | 0.03 | 27,020 | 0.02 | 2143 | 0.01 |
| Kidney cortex | 3429,797 | 1.09 | 1565,700 | 1.24 | 298,993 | 2.06 |
| Kidney medulla | 1283,496 | 0.41 | 494,144 | 0.39 | 86,467 | 0.60 |
| Liver | 2187,659 | 0.69 | 626,466 | 0.49 | 123,707 | 0.85 |
The mean (n = 2) radioactive content (dpm/g) of selected tissues in of C57BL/6J mice, 6, 24 and 72 h after a single 10 mg/kg oral dose of [14C]-fenclozic acid