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In vitro binding profile of GW405833
| Ki (nM) | rCB2/rCB1 Selectivity | Assay | Reference | ||||
|---|---|---|---|---|---|---|---|
| hCB1 | hCB2 | hCB2/hCB1 Selectivity | rCB1 | rCB2 | |||
| 4772 | 3.92 | 1217 | 273 | 3.6 | 76 | [3H] CP55,940 binding | Valenzano et al., 2005 |
| 282 | 7.62 | 37 | NA | 11.1 | NA | [3H] CP55,940 binding | Yao et al., 2008 |
| 1917 | 12 | 160 | NA | NA | NA | [3H] WIN55,212-2 binding | Gallant et al., 1996 |
NA, not available; hCB, human cannabinoid receptor; rCB, rat cannabinoid receptor.
